Mikael Bols

2019

Synthesis of Shld Derivatives, Their Binding to the Destabilizing Domain, and Influence on Protein Accumulation in Transgenic Plants

Jørgensen, F. P., Madsen, D., Meldal, M., Olsen, J. V., Petersen, M., Granhøj, J. & Bols, M., 23 May 2019, In: Journal of Medicinal Chemistry. 62, 10, p. 5191-5216 26 p.

Research output: Contribution to journal › Journal article › Research › peer-review

3 Citations (Scopus)

Zinc and Copper Complexes of Methylated Di- and Tetraaminocyclodextrins

Warren, J. & Bols, M., 7 Feb 2019, In: European Journal of Organic Chemistry. 2019, 5, p. 1083-1091 9 p.

Research output: Contribution to journal › Journal article › Research › peer-review

1 Citation (Scopus)

2018

An Inexpensive and Scalable Synthesis of Shld

Jørgensen, F. P. & Bols, M., 1 Jun 2018, In: Journal of Organic Chemistry. 83, 11, p. 6050-6055 6 p.

Research output: Contribution to journal › Journal article › Research › peer-review

7 Citations (Scopus)

2017

Artificial Metallooxidases from Cyclodextrin Diacids

Wang, B. & Bols, M., 4 Oct 2017, In: Chemistry: A European Journal. 23, 55, p. 13766-13775 10 p.

Research output: Contribution to journal › Journal article › Research › peer-review

19 Citations (Scopus)

Conformationally superarmed S-ethyl glycosyl donors as effective building blocks for chemoselective oligosaccharide synthesis in one pot

Bandara, M. D., Yasomanee, J. P., Rath, N. P., Pedersen, C. M., Bols, M. & Demchenko, A. V., 2017, In: Organic & Biomolecular Chemistry. 15, 3, p. 559-563 5 p.

Research output: Contribution to journal › Journal article › Research › peer-review

10 Citations (Scopus)

50 Downloads (Pure)

Determination of protonation states of iminosugar-enzyme complexes using photoinduced electron transfer

Wang, B., Olsen, J. I., Laursen, B. W., Poulsen, J. C. N. & Bols, M., 2017, In: Chemical Science. 8, 11, p. 7383-7393 11 p.

Research output: Contribution to journal › Journal article › Research › peer-review

7 Citations (Scopus)

78 Downloads (Pure)

Glycosyl Fluorides as Intermediates in BF₃ center dot OEt₂-Promoted Glycosylation with Trichloroacetimidates

Nielsen, M. M., A. Stougaard, B., Bols, M., Glibstrup, E. & Pedersen, C. M., 3 Mar 2017, In: European Journal of Organic Chemistry. 9, p. 1281-1284 4 p.

Research output: Contribution to journal › Journal article › Research › peer-review

8 Citations (Scopus)

On the nature of the electronic effect of multiple hydroxyl groups in the 6-membered ring - the effects are additive but steric hindrance plays a role too

Pedersen, C. M. & Bols, M., 2017, In: Organic & Biomolecular Chemistry. 15, 5, p. 1164-1173 10 p.

Research output: Contribution to journal › Journal article › Research › peer-review

7 Citations (Scopus)

97 Downloads (Pure)

Silyl-protective groups influencing the reactivity and selectivity in glycosylations

Bols, M. & Pedersen, C. M., 16 Jan 2017, In: Beilstein Journal of Organic Chemistry. 13, p. 93-105 13 p.

Research output: Contribution to journal › Journal article › Research › peer-review

35 Citations (Scopus)

155 Downloads (Pure)

2016

C-H functionalization on carbohydrates

Frihed, T. G., Bols, M. & Pedersen, C. M., Jun 2016, In: European Journal of Organic Chemistry. 2016, 16, p. 2740-2756 17 p.

Research output: Contribution to journal › Review › peer-review

13 Citations (Scopus)

Selenoureido-iminosugars: a new family of multitarget drugs

Olsen, J. I., Plata, G. B., Padrón, J. M., López, Ó., Bols, M. & Fernández-Bolaños, J. G., 2016, In: European Journal of Medicinal Chemistry. 123, p. 155-160 6 p.

Research output: Contribution to journal › Letter › peer-review

18 Citations (Scopus)

Super arming of a glycosyl donor using a molecular lever

Olsen, J. I., Kowalska, K., Pedersen, C. M. & Bols, M., 6 Jan 2016, In: Tetrahedron Letters. 57, 1, p. 35-38 4 p.

Research output: Contribution to journal › Letter › peer-review

4 Citations (Scopus)

2015

A fluorescence study of isofagomine protonation in β-glucosidase

Lindbäck, E. A., Laursen, B. W., Poulsen, J-C. N., Kilså, K., Pedersen, C. M. & Bols, M., 21 Jun 2015, In: Organic & Biomolecular Chemistry. 13, 23, p. 6562-6566 5 p.

Research output: Contribution to journal › Journal article › Research › peer-review

7 Citations (Scopus)

Exploring the relationship between the conformation and pK_a: can a pK_a value be used to determine the conformational equilibrium?

Olsen, J. I., Sauer, S. P. A., Pedersen, C. M. & Bols, M., 14 Mar 2015, In: Organic & Biomolecular Chemistry. 13, 10, p. 3116-3121 6 p.

Research output: Contribution to journal › Journal article › Research › peer-review

9 Citations (Scopus)

Mechanisms of glycosylation reactions studied by low-temperature nuclear magnetic resonance

Frihed, T., Bols, M. & Pedersen, C. M., 10 Jun 2015, In: Chemical Reviews. 115, 11, p. 4963-5013 51 p.

Research output: Contribution to journal › Review › peer-review

96 Citations (Scopus)

Synthesis of L-hexoses

Frihed, T., Bols, M. & Pedersen, C. M., 13 May 2015, In: Chemical Reviews. 115, 9, p. 3615-3676 62 p.

Research output: Contribution to journal › Review › peer-review

43 Citations (Scopus)

β-Mannosylation with 4,6-benzylidene protected mannosyl donors without preactivation

Heuckendorff, M., Bols, P. S., Barry, C. B., Frihed, T., Pedersen, C. M. & Bols, M., 13 Jul 2015, In: Chemical Communications. 51, 68, p. 13283-13285 3 p.

Research output: Contribution to journal › Journal article › Research › peer-review

29 Citations (Scopus)

2014

Cyclodextrin-based artificial oxidases with high rate accelerations and selectivity

Zhou, Y., Lindbäck, E. A., Pedersen, C. M. & Bols, M., 2014, In: Tetrahedron Letters. 55, 14, p. 2304-2307 4 p.

Research output: Contribution to journal › Journal article › Research › peer-review

9 Citations (Scopus)

Synthesis of all eight L-glycopyranosyl donors using C-H activation

Frihed, T., Pedersen, C. M. & Bols, M., 2014, In: Angewandte Chemie - International Edition. 53, 50, p. 13889-13893 5 p.

Research output: Contribution to journal › Journal article › Research › peer-review

22 Citations (Scopus)

Synthesis of all eight stereoisomeric 6-deoxy-l-hexopyranosyl donors - trends in using stereoselective reductions or mitsunobu epimerizations

Frihed, T., Pedersen, C. M. & Bols, M., 2014, In: European Journal of Organic Chemistry. 2014, 35, p. 7924-7939 16 p.

Research output: Contribution to journal › Journal article › Research › peer-review

21 Citations (Scopus)

Total synthesis of five lipoteichoic acids of Clostridium difficile

Hogendorf, W. F. J., Gisch, N., Schwudke, D., Heine, H., Bols, M. & Pedersen, C. M., 13 Oct 2014, In: Chemistry: A European Journal. 20, 42, p. 13511-13516 6 p.

Research output: Contribution to journal › Journal article › Research › peer-review

7 Citations (Scopus)

β-Selective mannosylation with a 4,6-silylene-tethered thiomannosyl donor

Heuckendorff, M., Bendix, J., Pedersen, C. M. & Bols, M., 21 Feb 2014, In: Organic Letters. 16, 4, p. 1116-9 4 p.

Research output: Contribution to journal › Journal article › Research › peer-review

48 Citations (Scopus)

2013

Artificial enzyme activity from cyclodextrins with cyanohydrins on the secondary rim

Zhou, Y., Pedersen, C. M. & Bols, M., 15 May 2013, In: Tetrahedron Letters. 54, 20, p. 2458-2461 4 p.

Research output: Contribution to journal › Journal article › Research › peer-review

9 Citations (Scopus)

Conformationally armed 3,6-tethered glycosyl donors: synthesis, conformation, reactivity, and selectivity

Heuckendorff, M., Pedersen, C. M. & Bols, M., 19 Jul 2013, In: Journal of Organic Chemistry. 78, 14, p. 7234-7248 15 p.

Research output: Contribution to journal › Journal article › Research › peer-review

45 Citations (Scopus)

Cyclodextrin-based artificial enzymes: synthesis and function

Pedersen, C. M. & Bols, M., 25 Oct 2013, Organic synthesis and molecular engineering. Brøndsted Nielsen, M. (ed.). Wiley, p. 305-332 28 p.

Research output: Chapter in Book/Report/Conference proceeding › Book chapter › Research › peer-review

5 Citations (Scopus)

Diethylsilane

Frihed, T., Bols, M. & Pedersen, C. M., 2013, e-EROS Encyclopedia of Reagents for Organic Synthesis. Fuchs, P. L. (ed.). Wiley

Research output: Chapter in Book/Report/Conference proceeding › Encyclopedia chapter › Research › peer-review

Enzyme inhibition by iminosugars: analysis and insight into the glycosidase-iminosugar dependency of pH

López, Ó., Qing, F-L., Pedersen, C. M. & Bols, M., 15 Aug 2013, In: Bioorganic & Medicinal Chemistry. 21, 16, p. 4755-4761 7 p.

Research output: Contribution to journal › Journal article › Research › peer-review

13 Citations (Scopus)

Influence of O6 in mannosylations using benzylidene protected donors: stereoelectronic or conformational effects?

Frihed, T., Walvoort, M. T. C., Codee, J. D. C., van der Marel, G. A., Bols, M. & Pedersen, C. M., 15 Mar 2013, In: Journal of Organic Chemistry. 78, 6, p. 2191-2205 15 p.

Research output: Contribution to journal › Journal article › Research › peer-review

34 Citations (Scopus)

Superarming of glycosyl donors by combined neighboring and conformational effects

Heuckendorff, M., Premathilake, H. D., Pornsuriyasak, P., Madsen, A. Ø., Pedersen, C. M., Bols, M. & Demchenko, A., 20 Sept 2013, In: Organic Letters. 15, 18, p. 4904-4907 4 p.

Research output: Contribution to journal › Journal article › Research › peer-review

19 Citations (Scopus)

Synthesis and thermotropic phase behavior of four glycoglycerolipids

Hogendorf, W. F. J., Jagalski, V., Günther-Pomorski, T., Bols, M., Cardenas Gomez, M. & Pedersen, C. M., Nov 2013, In: Molecules. 18, 11, p. 13546-13573 28 p.

Research output: Contribution to journal › Journal article › Research › peer-review

5 Citations (Scopus)

2012

Artificial enzymes based on cyclodextrin with phenol as the catalytic group

Lindbäck, E. A., Zhou, Y., Pedersen, C. M. & Bols, M., 12 Sept 2012, In: Tetrahedron Letters. 53, 37, p. 5023-5026 4 p.

Research output: Contribution to journal › Journal article › Research › peer-review

9 Citations (Scopus)

A uronic acid analogue of isofagomine lactam as a nanomolar glucuronidase inhibitor

Lindbäck, E. A., Zhou, Y., López, Ó., Fernández-Bolaños, J. G., Pedersen, C. M. & Bols, M., 18 Apr 2012, In: Tetrahedron Letters. 53, 16, p. 2045-2047 3 p.

Research output: Contribution to journal › Journal article › Research › peer-review

6 Citations (Scopus)

Conversion of D-glucose into 5-hydroxymethylfurfural (HMF) using zeolite in [Bmim]Cl or tetrabutylammonium chloride (TBAC)/CrCl₂

Jadhav, H. S., Taarning, E., Pedersen, C. M. & Bols, M., 22 Feb 2012, In: Tetrahedron Letters. 53, 8, p. 983-985 3 p.

Research output: Contribution to journal › Journal article › Research › peer-review

65 Citations (Scopus)

Easy access to L-Mannosides and L-Galactosides by using C-H activation of the corresponding 6-Deoxysugars

Frihed, T., Heuckendorff, M., Pedersen, C. M. & Bols, M., 3 Dec 2012, In: Angewandte Chemie International Edition. 51, 49, p. 12285–12288 4 p.

Research output: Contribution to journal › Journal article › Research › peer-review

33 Citations (Scopus)

Rhamnosylation: diastereoselectivity of conformationally armed donors

Heuckendorff, M., Pedersen, C. M. & Bols, M., 6 Jul 2012, In: Journal of Organic Chemistry. 77, 13, p. 5559-5568 10 p.

Research output: Contribution to journal › Journal article › Research › peer-review

28 Citations (Scopus)

Synthesis of cyclodextrins with carboxylic acids at the secondary rim and an evaluation of their properties as chemzymes for glycoside hydrolysis

Zhou, Y., Lindbäck, E. A., Marinescu-Pedersen, L. G., Pedersen, C. M. & Bols, M., Jul 2012, In: European Journal of Organic Chemistry. 2012, 21, p. 4063-4070 8 p.

Research output: Contribution to journal › Journal article › Research › peer-review

11 Citations (Scopus)

Synthesis of tin-containing cyclodextrins as potential enzyme models

Zhou, Y., Marinescu-Pedersen, L. G., Pedersen, C. M. & Bols, M., Nov 2012, In: European Journal of Organic Chemistry. 2012, 32, p. 6383-6389 7 p.

Research output: Contribution to journal › Journal article › Research › peer-review

9 Citations (Scopus)

Total synthesis of biologically active lipoteichoic acids

Pedersen, C. M., Bols, M. & Qiao, Y., 19 Dec 2012, In: ARKIVOC. 2013, 2, p. 249-275 27 p.

Research output: Contribution to journal › Journal article › Research › peer-review

1 Citation (Scopus)

Two diastereomeric artificial enzymes with different catalytic activity

Lindbäck, E. A., Zhou, Y., Pedersen, C. M. & Bols, M., Sept 2012, In: European Journal of Organic Chemistry. 2012, 27, p. 5366-5372 7 p.

Research output: Contribution to journal › Journal article › Research › peer-review

6 Citations (Scopus)

β-Cyclodextrin as a mimetic of the natural GFP-chromophore environment

Cacciarini, M., Nielsen, M. B., de Castro, E. M., Marinescu-Pedersen, L. G. & Bols, M., 22 Feb 2012, In: Tetrahedron Letters. 53, 8, p. 973-976 4 p.

Research output: Contribution to journal › Journal article › Research › peer-review

10 Citations (Scopus)

2011

3-Deoxyglucosone is an Intermediate in the Formation of Furfurals from D-Glucose

Jadhav, H. S., Pedersen, C. M., Sølling, T. I. & Bols, M., 22 Aug 2011, In: ChemSusChem. 4, p. 1049-1051

Research output: Contribution to journal › Journal article › Research › peer-review

60 Citations (Scopus)

An Isofagomine Analogue with an Amidine at the Pseudoanomeric Position

Lindbäck, E., López, Ó., Fernández-Bolaños, J. G., Sauer, S. P. A. & Bols, M., 3 Jun 2011, In: Organic Letters. 13, 11, p. 2908-2911

Research output: Contribution to journal › Journal article › Research › peer-review

13 Citations (Scopus)

A study of anhydrocelluloses - Is a cellulose structure with residues in a 1C4-conformation more prone to hydrolysis?

Jadhav, V., Pedersen, C. M. & Bols, M., 7 Nov 2011, In: Organic & Biomolecular Chemistry. 9, 21, p. 7525-7534

Research output: Contribution to journal › Journal article › Research › peer-review

10 Citations (Scopus)

Cyclodextrin Ketones with the Catalytic Group at the Secondary Rim and Their Effectiveness in Enzyme-Like Epoxidation of Stilbenes

Fenger, T. H., Marinescu-Pedersen, L. G. & Bols, M., Apr 2011, In: European Journal of Organic Chemistry. p. 2339-2345 7 p.

Research output: Contribution to journal › Journal article › Research › peer-review

16 Citations (Scopus)

Direct Experimental Evidence for the High Chemical Reactivity of a- and ß-Xylopyranosides Adopting a 2,5B Conformation in Glycosyl Transfer

Amorim, L., Marcelo, F., Rousseau, C. A. R., Nieto, L., Jimenez-Barbero, J., Marrot, J., Rauter, A. P., Sollogoub, M., Bols, M. & Bleriot, Y., 2011, In: Chemistry: A European Journal. 17, p. 7345–7356

Research output: Contribution to journal › Journal article › Research › peer-review

Glycosyl Donors in ‘Unusual’ Conformations – Influence on Reactivity and Selectivity.

Bols, M. & Pedersen, C. M., Jan 2011, In: Proceedings of the Russian Academy of Sciences.

Research output: Contribution to journal › Literature review › Research › peer-review

52 Citations (Scopus)

Quantifying the Electronic Effects of Carbohydrate Hydroxy Groups by Using Aminosugar Models

Pedersen, C. M., Olsen, J., Brka, A. & Bols, M., 14 Jun 2011, In: Chemistry: A European Journal. 17, 25, p. 7080-7086

Research output: Contribution to journal › Journal article › Research › peer-review

37 Citations (Scopus)

Recognition of Peptides by Cyclodextrin Trimers

Christensen, H. S., Sigurdskjold, B., Frihed, T., Marinescu-Pedersen, L. G., Pedersen, C. M. & Bols, M., Sept 2011, In: European Journal of Organic Chemistry. 27, p. 5279-5290

Research output: Contribution to journal › Journal article › Research › peer-review

21 Citations (Scopus)

Regioselective difunctionalization of cyclodextrins.

Petrillo, M., Marinescu-Pedersen, L. G. & Bols, M., Apr 2011, In: Journal of Inclusion Phenomena and Macrocyclic Chemistry. p. 425-431 7 p.

Research output: Contribution to journal › Journal article › Research › peer-review

6 Citations (Scopus)

Simple cyclodextrin aldehydes as excellent artificial oxidases.

Fenger, T. H. & Bols, M., Apr 2011, In: Journal of Inclusion Phenomena and Macrocyclic Chemistry. 69, 3-4, p. 397-402 6 p.

Research output: Contribution to journal › Journal article › Research › peer-review

13 Citations (Scopus)

Mikael Bols

Research output

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