Partial agonism and antagonism of the ionotropic glutamate receptor iGLuR5: Structures of the ligand-bining core in complex with domoic acid and 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid

Helle Hald; Peter Naur; Darryl Scott Pickering; Desiree Sprogøe; Ulf Madsen; Daniel B. Timmermann; Philip K. Ahring; Tommy Liljefors; Arne Schousboe; Jan Egebjerg; Michael Gajhede; Jette Sandholm Jensen Kastrup

doi:10.1074/jbc.M700137200

Partial agonism and antagonism of the ionotropic glutamate receptor iGLuR5: Structures of the ligand-bining core in complex with domoic acid and 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid

Helle Hald, Peter Naur, Darryl Scott Pickering, Desiree Sprogøe, Ulf Madsen, Daniel B. Timmermann, Philip K. Ahring, Tommy Liljefors, Arne Schousboe, Jan Egebjerg, Michael Gajhede, Jette Sandholm Jensen Kastrup

39 Citations (Scopus)

Original language	English
Journal	Journal of Biological Chemistry
Volume	282
Issue number	35
Pages (from-to)	25726-25736
ISSN	0021-9258
DOIs	https://doi.org/10.1074/jbc.M700137200
Publication status	Published - 2007

Keywords

Former Faculty of Pharmaceutical Sciences

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10.1074/jbc.M700137200

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Hald, H., Naur, P., Pickering, D. S., Sprogøe, D., Madsen, U., Timmermann, D. B., Ahring, P. K., Liljefors, T., Schousboe, A., Egebjerg, J., Gajhede, M., & Kastrup, J. S. J. (2007). Partial agonism and antagonism of the ionotropic glutamate receptor iGLuR5: Structures of the ligand-bining core in complex with domoic acid and 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid. Journal of Biological Chemistry, 282(35), 25726-25736. https://doi.org/10.1074/jbc.M700137200

Partial agonism and antagonism of the ionotropic glutamate receptor iGLuR5 : Structures of the ligand-bining core in complex with domoic acid and 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid. / Hald, Helle; Naur, Peter; Pickering, Darryl Scott et al.

In: Journal of Biological Chemistry, Vol. 282, No. 35, 2007, p. 25726-25736.

Research output: Contribution to journal › Journal article › Research › peer-review

Hald, H, Naur, P, Pickering, DS, Sprogøe, D, Madsen, U, Timmermann, DB, Ahring, PK, Liljefors, T, Schousboe, A, Egebjerg, J, Gajhede, M & Kastrup, JSJ 2007, 'Partial agonism and antagonism of the ionotropic glutamate receptor iGLuR5: Structures of the ligand-bining core in complex with domoic acid and 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid', Journal of Biological Chemistry, vol. 282, no. 35, pp. 25726-25736. https://doi.org/10.1074/jbc.M700137200

Hald H, Naur P, Pickering DS, Sprogøe D, Madsen U, Timmermann DB et al. Partial agonism and antagonism of the ionotropic glutamate receptor iGLuR5: Structures of the ligand-bining core in complex with domoic acid and 2-amino-3-[5-tert-butyl-3-(phosphonomethoxy)-4-isoxazolyl]propionic acid. Journal of Biological Chemistry. 2007;282(35):25726-25736. doi: 10.1074/jbc.M700137200

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AU - Gajhede, Michael

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