Synthesis, radiolabeling and in vivo evaluation of [C-11](R)-1-[4-[2-(4-methoxyphenyl)phenyl piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT7 receptor

Hanne D. Hansen; Enza Lacivita; Pantaleo Di Pilato; Matthias Manfred Herth; Szabolcs Lehel; Anders Ettrup; Valdemar L. Andersen; Agnete Dyssegaard; Paola De Giorgio; Roberto Perrone; Francesco Berardi; Nicola Antonio Colabufo; Mauro Niso; Gitte M. Knudsen; Marcello Leopoldo

doi:10.1016/j.ejmech.2014.03.066

Synthesis, radiolabeling and in vivo evaluation of [C-11](R)-1-[4-[2-(4-methoxyphenyl)phenyl piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT7 receptor

Hanne D. Hansen, Enza Lacivita, Pantaleo Di Pilato, Matthias Manfred Herth, Szabolcs Lehel, Anders Ettrup, Valdemar L. Andersen, Agnete Dyssegaard, Paola De Giorgio, Roberto Perrone, Francesco Berardi, Nicola Antonio Colabufo, Mauro Niso, Gitte M. Knudsen, Marcello Leopoldo

16 Citationer (Scopus)

Originalsprog	Engelsk
Tidsskrift	European Journal of Medicinal Chemistry
Vol/bind	79
Sider (fra-til)	152-163
Antal sider	12
ISSN	0223-5234
DOI	https://doi.org/10.1016/j.ejmech.2014.03.066
Status	Udgivet - 22 maj 2014

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10.1016/j.ejmech.2014.03.066

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Hansen, H. D., Lacivita, E., Di Pilato, P., Herth, M. M., Lehel, S., Ettrup, A., Andersen, V. L., Dyssegaard, A., De Giorgio, P., Perrone, R., Berardi, F., Colabufo, N. A., Niso, M., Knudsen, G. M., & Leopoldo, M. (2014). Synthesis, radiolabeling and in vivo evaluation of [C-11](R)-1-[4-[2-(4-methoxyphenyl)phenyl piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT7 receptor. European Journal of Medicinal Chemistry, 79, 152-163. https://doi.org/10.1016/j.ejmech.2014.03.066

Synthesis, radiolabeling and in vivo evaluation of [C-11](R)-1-[4-[2-(4-methoxyphenyl)phenyl piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT7 receptor. / Hansen, Hanne D.; Lacivita, Enza; Di Pilato, Pantaleo et al.
I: European Journal of Medicinal Chemistry, Bind 79, 22.05.2014, s. 152-163.

Publikation: Bidrag til tidsskrift › Tidsskriftartikel › Forskning › peer review

Hansen, HD, Lacivita, E, Di Pilato, P, Herth, MM, Lehel, S, Ettrup, A, Andersen, VL, Dyssegaard, A, De Giorgio, P, Perrone, R, Berardi, F, Colabufo, NA, Niso, M, Knudsen, GM & Leopoldo, M 2014, 'Synthesis, radiolabeling and in vivo evaluation of [C-11](R)-1-[4-[2-(4-methoxyphenyl)phenyl piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT7 receptor', European Journal of Medicinal Chemistry, bind 79, s. 152-163. https://doi.org/10.1016/j.ejmech.2014.03.066

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title = "Synthesis, radiolabeling and in vivo evaluation of [C-11](R)-1-[4-[2-(4-methoxyphenyl)phenyl piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT7 receptor",

keywords = "5-HT7 receptor, PET, Radioligand, Arylpiperazine, SB-269970",

author = "Hansen, {Hanne D.} and Enza Lacivita and {Di Pilato}, Pantaleo and Herth, {Matthias Manfred} and Szabolcs Lehel and Anders Ettrup and Andersen, {Valdemar L.} and Agnete Dyssegaard and {De Giorgio}, Paola and Roberto Perrone and Francesco Berardi and Colabufo, {Nicola Antonio} and Mauro Niso and Knudsen, {Gitte M.} and Marcello Leopoldo",

year = "2014",

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doi = "10.1016/j.ejmech.2014.03.066",

language = "English",

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T1 - Synthesis, radiolabeling and in vivo evaluation of [C-11](R)-1-[4-[2-(4-methoxyphenyl)phenyl piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT7 receptor

AU - Hansen, Hanne D.

AU - Lacivita, Enza

AU - Di Pilato, Pantaleo

AU - Herth, Matthias Manfred

AU - Lehel, Szabolcs

AU - Ettrup, Anders

AU - Andersen, Valdemar L.

AU - Dyssegaard, Agnete

AU - De Giorgio, Paola

AU - Perrone, Roberto

AU - Berardi, Francesco

AU - Colabufo, Nicola Antonio

AU - Niso, Mauro

AU - Knudsen, Gitte M.

AU - Leopoldo, Marcello

PY - 2014/5/22

Y1 - 2014/5/22

KW - 5-HT7 receptor

KW - PET

KW - Radioligand

KW - Arylpiperazine

KW - SB-269970

U2 - 10.1016/j.ejmech.2014.03.066

DO - 10.1016/j.ejmech.2014.03.066

M3 - Journal article

C2 - 24732791

SN - 0223-5234

VL - 79

SP - 152

EP - 163

JO - European Journal of Medicinal Chemistry

JF - European Journal of Medicinal Chemistry

ER -

Synthesis, radiolabeling and in vivo evaluation of [C-11](R)-1-[4-[2-(4-methoxyphenyl)phenyl piperazin-1-yl]-3-(2-pyrazinyloxy)-2-propanol, a potential PET radioligand for the 5-HT7 receptor

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