Design and synthesis of a stable oxidized phospholipid mimic with specific binding recognition for macrophage scavenger receptors

William W Turner, Karsten Hartvigsen, Agnes Boullier, Erica N Montano, Joseph L Witztum, Michael S VanNieuwenhze

8 Citationer (Scopus)

Abstract

Macrophage scavenger receptors appear to play a major role in the clearance of oxidized phospholipid (OxPL) products. Discrete peptide-phospholipid conjugates with the phosphatidylcholine headgroup have been shown to exhibit binding affinity for these receptors. We report the preparation of a water-soluble, stable peptide-phospholipid conjugate (9) that possesses the necessary physical properties to enable more detailed study of the role(s) of OxPL in metabolic disease.
OriginalsprogEngelsk
TidsskriftJournal of Medicinal Chemistry
Vol/bind55
Udgave nummer18
Sider (fra-til)8178-82
Antal sider5
ISSN0022-2623
DOI
StatusUdgivet - 27 sep. 2012

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